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The O
Lung cancer and matrix metalloproteinases inhibitors of polyphenols from Selaginella tamariscina with suppression activity of migration PMID 29921475
(S)
Methyl (E)
Cardiovascular effects of griseofulvin PMID 5652459
BCI
(9E,12E)
Effect of HM30181 mesylate salt
Chromatographic Evaluation and Characterization of Constituents of Sunflower Seed Extract Used as Food Additives PMID 38233137
PRMT5
Transport of Adoptive Cell Transfers With Magnetic Helical Microrobots PMID 40911713
Panclicins, novel pancreatic lipase inhibitors. II. Structural elucidation PMID 7844032
lac Repressor
Danicamtiv 1970972
NAD+ Kinase as a Therapeutic Target in Cancer PMID 27582489
血小板衍生生长因子 D（PDGFD）基因
Oxonol VI 64724
exo
Synthesis of novel trifluoromethyl substituted furo[2,3
Synthesis and biological evaluation of polymethoxylated 4
Design, synthesis and biological evaluation of novel benzocoumarin derivatives as potent inhibitors of MAO
Benzoic acid allopyranosides from the bark of Pseudolarix kaempferi PMID 16808935
(Rac)
Dioxybenzone (Standard)
1,1
p
Lancifodilactone C 663176
Rapid synthesis of 4
Synthesis and biological evaluation of 1
NADH dehydrogenase.
inorganic chemical compound
Terpenes from Copaifera demonstrated in vitro antiparasitic and synergic activity PMID 22440015
Jietacins, azoxy natural products, as novel NF
β
胰岛素样生长因子结合蛋白 3（IGFBP3）基因
Barakol 24506
Tryptophan
Anti
Omecamtiv mecarbil
跨膜 4 L 6 家族成员 19（TM4SF19）基因
Aethimidinum
Boc
L
Identification of 3H
Cystocholic acid 73386
Methyl trioctyl ammonium
Naphthalene/quinoline amides and sulfonylureas as potent and selective antagonists of the EP4 receptor PMID 21215624
Investigation of stability of selective androgen receptor modulators in urine PMID 32401172
R916562 1037798
羊毛甾醇合酶（LSS）基因
Zaldaride maleate 109826
Chitosan
p
Cilengitide sensitivity is predicted by overall integrin expression in breast cancer PMID 39707454
Sorivudine and 5
达兹托肽, 达多肽
Depudecin a novel compound inducing the flat phenotype of NIH3T3 cells doubly transformed by ras
Blockade of JAK2 protects mice against hypoxia
Brassinin 105748
CD39 improves survival in microbial sepsis by attenuating systemic inflammation PMID 25318479
AMPK activator
Chalkone Glycosidenatural
RAB32，RAS 致癌基因家族成员（RAB32）基因
Vgll4
MU380 2109805
Ascorutin
Insertion and organization within membranes of the delta
The P38MAPK Pathway Mediates the Destruction of the Blood
The antiviral activity of caprochlorone PMID 6027546
IRE1α
Exploration and validation of therapeutic molecules for rheumatoid arthritis based on ferroptosis
Pheromone biosynthesis activating neuropeptide (PBAN) regulatory role and mode of action PMID 18495120
Identification of dibucaine derivatives as novel potent enterovirus 2C helicase inhibitors In vitro, in vivo, and combination therapy study PMID 32619885
Chlovalicin 179799
Isoallolithocholic acid 2276
丝氨酸/苏氨酸激酶 16（STK16）基因
Akt1
Ebrotidine
In vivo trypanosomicidal activity of imidazole
SREBF1 facilitates pathological retinal neovascularization by reprogramming the fatty acid metabolism of endothelial cells PMID 39800283
ACC1
2,4
L
Nortropinone hydrochloride 25602
The Indenoisoquinoline LMP517 A Novel Antitumor Agent Targeting both TOP1 and TOP2 PMID 32430490
Prozac (fluoxetine, Lilly 110140), the first selective serotonin uptake inhibitor and an antidepressant drug twenty years since its first publication PMID 7623609
Acetylvaline (Standard)
4,6
1,3
镰孢菌素 B
3
Heme oxygenase
Fosciclopirox disodium 1380539
ZSH
Neuropeptide Y (13
Cyclic somatostatin
N
N
核受体亚家族 3 C 组成员 2（NR3C2）基因
DD0
Pipermethystine
A 419259 trihydrochloride (RK 20449 trihydrochloride)
Structure
Induction of apoptosis and antiproliferative activity of naringenin in human epidermoid carcinoma cell through ROS generation and cell cycle arrest PMID 25330158
TMX
BRD4 Inhibitor
Peluntamig (PT
idasanutlin
Etiocholanolone (5β
DHC
PSI
腾冲过路黄提取物 (Lysimachia tengyuehensis Hand.
ODN 1018 (1018 ISS)
TGP
metabolic disorder
Structure
BChE
Avermectin induces photoreceptor functional impairment and color vision deficits in zebrafish (Danio rerio) PMID 40174454
Dodecamethylpentasiloxane 141
GTSE1
FR264205
Targeting energy metabolic and oncogenic signaling pathways in triple
dAURK
AZD4747
SCH 486757
NRCMs
PRN1371
TMEM160 inhibits KEAP1 to suppress ferroptosis and induce chemoresistance in gastric cancer PMID 40223081
Ponasterone A 13408
Group II metabotropic glutamate receptor agonist prodrugs LY2979165 and LY2140023 attenuate the functional imaging response to ketamine in healthy subjects PMID 29564482
ANVS 401
Platycodin D 58479
BAY
Coenzyme Q10 prevents RANKL
RAW264.7 cells
(Sar1,Ile4,8)
Izonsteride
Using siRNA
F14679
ABCC1 蛋白, Human (His)
Impedance
MCE
Modified (2'
INCB18424
SLAMF6 蛋白, Human (HEK293, His
3,5,6,7,8,3',4'
cyclo
Dynamic assessment of PI4P metabolism using split GFP based sensors PMID 40841827
Efficacy of the MCHR1 antagonist N
3
AQX
MCE
尤尼妥单抗
1,4
(S)
AZ876
Disubstituted piperidines as potent orexin (hypocretin) receptor antagonists PMID 22617492
Indazole
The CXC chemokine cCAF stimulates precocious deposition of ECM molecules by wound fibroblasts, accelerating development of granulation tissue PMID 12057014
Cyclin dependent kinase (CDK) inhibitors as anticancer drugs Recent advances (2015
Cholesterol neutralized vemurafenib treatment by promoting melanoma stem
hypomethylating
ODN 1668
雷琐酚
A
N,N'
Firsocostat (ND
S49076 hydrochloride
LP99 Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor PMID 25864491
Novel allosteric glutaminase 1 inhibitors with macrocyclic structure activity relationship analysis PMID 36038117
9(Z),12(Z)
CEACAM5 蛋白, Human (HEK293, Fc)
Sofosbuvir impurity C (索非布韦杂质C)
Development and Characterization of a Fluorescent Probe for GLS1 and the Application for High
雷琐酚
Structure
XmAb
hypomethylating
Delivery of insulin
PTP4A2 蛋白, Human (GST)
CFM
Desamino(D
Crocin II (Standard)
Sulfo
Mesenchymal stem cells
Anti
Picrotoxinin
α
Lysimachigenoside C
SM1044
Ubiquinone Q9
S1P1 agonist 5
Maackia Amurensis Lectin I (Fluorescein) (MAL I (Fluorescein))
Synthesis of N
Oseltamivir
D
半乳糖
3,5,6
Campathecin
Pseudolaroside B
M1069
Cathepsin L1 蛋白, Mouse (HEK293, His)
Cy7.5 HA (MW 10000) (Cy7.5 标记 透明质酸 (MW 10000))
DLC27
2
FT 001
Dexamethasone palmitate (Standard)
CGP 062464
Dihydrobaicalein
Novel amino substituted tetracyclic imidazo[4,5
Discovery of a Thiadiazole
Bim 抗体 (YA582)（Bim Antibody (YA582)）
(5R)
Discovery of IPN60090, a Clinical Stage Selective Glutaminase
Sarracenin
A series of novel aryl
Zinpyr
Synthesis and evaluation of bisbenzylidenedioxotetrahydrothiopranones as activators of endoplasmic reticulum (ER) stress signaling pathways and apoptotic cell death in acute promyelocytic leukemic cells PMID 24960549
4
Oseltamivir
聚合酶链式反应
Methyl
Discovery and development of novel pyrimidine and pyrazolo/thieno
Birc2
Janelia Fluor® 549 TFA (JF549 TFA)
2'
Aleuria Aurantia Lectin (Agarose) (AAL (Agarose))
Bis(trimethylsilyl)acetylene 14630
Sevoflurane acts as an antidepressant by suppression of GluN2D
New crinine
MCE
Dihydrostilbenes and diarylpropanes Synthesis and in vitro pharmacological evaluation as potent nitric oxide production inhibition agents PMID 27777005
Fluorinated rhodacyanine (SJL
Acylated phenylethanoid oligoglycosides with hepatoprotective activity from the desert plant Cistanche tubulosa PMID 20159656
Oseltamivir
Discovery of potent, isoform
DL
KRAS
Oseltamivir
Adamantane 11
JNJ
Endoxifen hydrochloride 1197194
KTX
Flavaglines as potent anticancer and cytoprotective agents PMID 23072299
Wnt3a 抗体（Wnt3a Antibody）
Cyclopeptides from the Sponge Stylissa flabelliformis PMID 29893558
Discovery of a Series of 2'
Dissymmetric pyridyl
Design and synthesis of thiourea derivatives containing a benzo[5,6]cyclohepta[1,2
A novel class of thiosemicarbazones show multi
Gastric ulcer
Towards a new combination therapy for tuberculosis with next generation benzothiazinones PMID 24500695
OX1a 136340
Oseltamivir
Human
Multi
Selective cytotoxicity of oxysterols through structural modulation on rings A and B. Synthesis, in vitro evaluation, and SAR PMID 21797280
Improved correction of F508del
Leptin (116
Synthesis and anti
E3 ubiquitination ligase XIAP lightens diabetes
Discovery of a Novel, Highly Potent, and Selective Thieno[3,2
CD158z/KIR3DL3
Design, synthesis and biological evaluation of [1,2,4]triazolo[1,5
KRAS
Meclizine dihydrochloride
Synthesis of novel tricyclic chromenone
Nurandociguatum (Nurandociguat)
Structural development of a type
FAK inhibitor
BMS
Discovery of Dual CDK6/PIM1 Inhibitors with a Novel Structure, High Potency, and Favorable Druggability for the Treatment of Acute Myeloid Leukemia PMID 34958208
Discovery of novel glutaminase 1 allosteric inhibitor with 4
Furagin (Furazidine，呋喃烯啶)
The discovery and optimization of novel dual inhibitors of topoisomerase II and histone deacetylase PMID 24095018
CD25 抗体 (YA5368)（CD25 Antibody (YA5368)）
Fas 激活的丝氨酸/苏氨酸激酶（FASTK）基因
三肽基肽酶 2（TPP2）基因
Oxidation of phenethylamine derivatives by cytochrome P450 2D6 the issue of substrate protonation in binding and catalysis PMID 11714275
Glucosamine
hsa
6
英克司兰钠
NBI
Structure
Gdf15
Hexamethylene dibromide
Mutagenesis studies of the 14 Å internal cavity of histone deacetylase 1 insights toward the acetate
Rubriflorin B 835875
Identification of Pyruvate Carboxylase as the Cellular Target of Natural Bibenzyls with Potent Anticancer Activity against Hepatocellular Carcinoma via Metabolic Reprogramming PMID 34931827
Cafestol palmitate
A novel small molecule chaperone of rod opsin and its potential therapy for retinal degeneration PMID 29773803
Human leukocyte immunoglobulin (Ig)
LAQ 824
Kinetic and structural insights into the binding of histone deacetylase 1 and 2 (HDAC1, 2) inhibitors PMID 27377864
Exploring the Implication of DDX3X in DENV Infection Discovery of the First
Total Synthesis and Biological Studies of TMC
FITC
COX
TASK Channels Pharmacology New Challenges in Drug Design PMID 31260312
Synthesis and Biological Activity of Triterpene
The discovery of N
The kinetics of cytokine gene expression in the thyroids of mice developing granulomatous experimental autoimmune thyroiditis PMID 9878080
Long intergenic non
Cytotoxic triterpene dilactones from the stems of Kadsura ananosma PMID 20025236
N
UMB298
NS5 RdRp
The discovery of indole full agonists of the neurotensin receptor 1 (NTSR1) PMID 24997685
Filricianine
Metabolomic analysis revealed glycylglycine accumulation in astrocytes after methionine enkephalin administration exhibiting neuron protective effects PMID 26163404
金合欢提取物 (Acacia farnesiana (Linn.) Willd.)
A novel protein CYTB
Sergliflozin
Ruxolitinib Alleviates Inflammation and Fortifies Skin Barrier Function Through Dampening IL
Pyridalyl 179101
Aromatic beta
HER4 蛋白, Human (HEK293, His
Design and evaluation of novel glutaminase inhibitors PMID 26988803
Identification of steroid
Thymine (胸腺嘧啶)
Ostruthin 148
Small
TREM2 deficiency in microglia accelerates photoreceptor cell death and immune cell infiltration following retinal detachment PMID 36977680
Antiplatelet aggregation principles of Dendrobium loddigesii PMID 7798962
Perfluorodecyl bromide 307
Fragment
Cyclooxygenase
Synthesis and evaluation of a series of benzothiophene acrylonitrile analogs as anticancer agents PMID 23956835
2
A431 cells
Hdac8 Mouse Pre
Methylophiopogonone A (Standard)
IL
Discovery and Synthesis of a Phosphoramidate Prodrug of a Pyrrolo[2,1
N
Discovery of a Potent and Selective TRPC5 Inhibitor, Efficacious in a Focal Segmental Glomerulosclerosis Model PMID 31749913
TAK
SMARCA2/4
Intermittent theta
In search of a cytostatic agent derived from the alkaloid lycorine synthesis and growth inhibitory properties of lycorine derivatives PMID 22019045
Sesquiterpenes from the roots of Lindera strychnifolia with inhibitory effects on nitric oxide production in RAW 264.7 cells PMID 27634197
川牛膝提取物 (Cyathula officinalis Kuan)
(tert
NXE 0041178
Water
(±)
CEBP delta/CEBPD 蛋白, Human (His
Specnuezhenide mitigates tunicamycin
Antitumor agents 7. Synthesis, antiproliferative activity and molecular modeling of new l
Potent naphthoquinones against antimony
Dealanylalahopcin
NR3C1 Human Pre
Meclofenamic acid
PMH
Cytotoxic alkaloids from the whole plants of Zephyranthes candida PMID 23190013
HuM291
AJH836
Phenolic compounds from Caesalpinia sappan heartwood and their anti
Eno1 Rat Pre
A Bioreductive Prodrug of Cucurbitacin B Significantly Inhibits Tumor Growth in the 4T1 Xenograft Mice Model PMID 31620225
Semisynthetic studies identify mitochondria poisons from botanical dietary supplements
EF24 induces G2/M arrest and apoptosis in cisplatin
cGAS/STING signalling in macrophages aggravates obliterative bronchiolitis via an IFN
Diclofenac Sodium Restores the Sensitivity of Colistin
Synthesis and anti
Discovery, design and synthesis of Y
Hexamethylene dibromide
Nonhydrolyzable ATP analog 5'
LFS
Glucosamine
An Alkyne
Binding to an Unusual Inactive Kinase Conformation by Highly Selective Inhibitors of Inositol
Klk1
SWTX
Methyl 2
furan
ECIN 66160
Small Molecule Mitochondrial Uncouplers and Their Therapeutic Potential PMID 29156129
FAAH
Diethyl 3
Synthesis and biological evaluation of cyanoguanidine derivatives of loratadine PMID 22959205
Discovery of isoindoline and tetrahydroisoquinoline derivatives as potent, selective PPARδ agonists PMID 21094606
Lenalidomide 4'
(4
Amaryllidaceae alkaloids belonging to different structural subgroups display activity against apoptosis
Liposomal formulation of retinoids designed for enzyme triggered release PMID 20405849
Genkwanin reduces airway epithelial cell ferroptosis and alleviates asthma symptoms in mice PMID 41046685
Lead Optimization of Benzoxazolone Carboxamides as Orally Bioavailable and CNS Penetrant Acid Ceramidase Inhibitors PMID 32176488
Discovery of Competitive and Noncompetitive Ligands of the Organic Cation Transporter 1 (OCT1; SLC22A1) PMID 28230985
Kisspeptin
DABCYL
Apt
Discovery of AMG 232, a potent, selective, and orally bioavailable MDM2
Cytotoxic steroidal alkaloids from Kibatalia laurifolia PMID 21443172
3& 039;
Boc
ELQ
aggression
2
Dual Targeting of BRAF and mTOR Signaling in Melanoma Cells with Pyridinyl Imidazole Compounds PMID 32531927
SF3B1
Dimethyl
Guajadial F 1529775
Challenges in the development of an M4 PAM in vivo tool compound The discovery of VU0467154 and unexpected DMPK profiles of close analogs PMID 27939174
Antiprotozoal Sesquiterpene Lactones and Other Constituents from Tarchonanthus camphoratus and Schkuhria pinnata PMID 29244495
Dextran blue (MW 2000000)
Review article metoclopramide and tardive dyskinesia PMID 19886950
Anti
Rational modifications, synthesis and biological evaluation of new potential antivirals for RSV designed to target the M2
Spirobisnaphthalenes and lactones from the seeds of Strychnos angustiflora with potential anti
Design, synthesis and preclinical evaluation of NRC
Anti
匹伐他汀钙(Standard)
KGF
PIP4P1 Human Pre
Human IgG1 (F405L) kappa, Isotype Control
Sustained
Effect of gestational age and hypoxia on activity of ribonucleic acid polymerase in fetal guinea pig brain PMID 11262481
PPZ
Discovery of 4'
4
On the vasoprotective mechanisms underlying novel β
β
Studies towards the conception of new selective PPARbeta/delta ligands PMID 16797985
Ramatroban
N
The toxic mechanism and metabolic effects of atractyloside in precision
C12
Synthesis of C2
Aminomethylation of heliomycin Preparation and anticancer characterization of the first series of semi
Verubecestat (Standard)
Sesquiterpene Lactones from Artemisia argyi Absolute Configuration and Immunosuppressant Activity PMID 31181920
4
KO 947
BRL 37344
(2S,7aR)
Red cochineal dye (carminic Acid) its role in nature PMID 17779027
Ro 2
(R)
Gd
Homovanillic acid
3
头孢磺吡酮(Standard)
Guaiphenesin(Standard)
那美芦单抗
hydrolyze
Effects of substance P and substance P
GSK
TK
Doxorubicin and Aclarubicin Shuffling Anthracycline Glycans for Improved Anticancer Agents PMID 33064004
A comparison of the beta
sigma receptors
Design of isoform
Tricin (Standard)
Sofosbuvir
PNU
Rhazinilam and quebrachamine derivatives from Yunnan Kopsia arborea PMID 19133778
2
Thalidomide
Aldehyde dehydrogenases
BPU
Design, in silico prioritization and biological profiling of apoptosis
Discovery of pyrimidine nucleoside dual prodrugs and pyrazine nucleosides as novel anti
Dalosirvat (SM
Olorigliflozin
L
VISTA is an immune checkpoint molecule for human T cells PMID 24691993
Plant isoquinoline alkaloids Advances in the chemistry and biology of berberine PMID 34536668
Elafibranor, an Agonist of the Peroxisome Proliferator
Remogliflozin (Remogliflozin A)
Evaluation of THP
Flavokawain A (Standard) (卡瓦胡椒素A (Standard))
Discovery of non
Moscatilin Ameliorates Tau Phosphorylation and Cognitive Deficits in Alzheimer's Disease Models PMID 31291099
Nintedanib impurity 4
4
AH
IC
NBC 19
SF 22
Verekitug
JA2131
3
pyrimidine piperazine
biliary epithelial cells
3,4
Dinoprost
Pimavanserin hemitartrate (Standard)
Dioscorea collettii
LacCer
ULK1 Knockout Exacerbates Ischemia
Solution structure of amyloid beta
Ghrelin improves endothelial function and reduces blood pressure in Ang II
N
ET receptor antagonist 2
4
CN128 hydrochloride (CN328)
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